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位点连接药物设计法
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位点连接药物设计法
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site point connection-based drug design
位点连接药物设计法
根据位点特征和位置,在靶标活性口袋中放入合适的配体分子片段的方法。位点就是在活性口袋中能与靶标的化学特征相匹配的结构模式。
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