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靶标确证
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target validation
靶标确证
在发现活性小分子化合物潜在靶标蛋白的基础上,采取生物化学、分子生物学、生物物理、化学蛋白质组学等方法,结合体外和体内分析,证实活性小分子与靶蛋白的直接作用介导了活性小分子生物学效应的方法。
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