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metabolic antagonism
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metabolic antagonism
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代谢拮抗
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metabolic antagonism
代谢拮抗
设计与生物体内基本代谢物的结构相似的化合物,使之竞争性地与特定的酶作用,干扰基本代谢物的被利用,从而干扰生物大分子的合成;或以伪代谢物的身份掺入生物大分子的合成中,形成伪生物大分子,导致致死合成,从而影响细胞的生长。
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